ICOS-20, 20th International Conference on Organic Synthesis
 
 
Friday, 20 October 2017
 
 
Detailed program

 

Sunday, 29 June 2014

12:00 - 17:00 Registration
13:30 - 16:30 Unique tour to Egis
17:00 - 17:30 Opening ceremony - Chair: Péter Mátyus
17:30 - 18:30 Chair: Eusebio Juaristi
PL-1 Lutz F. Tietze, Germany
The Concept of Domino Reactions: An Approach to the Ideal Synthesis
18:30 - 19:30 PL-2 Jay Siegel, China
Cationic Organisilanes and C-F Activation
19:30 - 21:30 Welcome Party
 

Monday, 30 June 2014

07:30 - 08:45 Registration

Chair: Mark A. Rizzacasa
08:45 - 09:45 PL-3 Margaret A Brimble, New Zealand
Synthesis of Natural Products Containing Aromatic Spiroketals
09:45 - 10:15 IL-1 Tohru Fukuyama, Japan
Synthetic Studies on (–)-Oxycodone
10:15 - 10:45 IL-2 Stephen Kent, United States
Total Chemical Synthesis of Proteins, the Natural Products of the 21st Century
10:45 - 11:15 Coffee Break

Short Oral Presentations

Session I

Chair: Kevin Booker-Milburn
11:15 - 11:30 L-1 Takanori Shibata, Japan
Enantioselective Synthesis of Paracyclophanes and Their Use as Chiral Ligands in Asymmetric Coupling
11:30 - 11:45 L-2 Okiko Miyata, Japan
Sequential Retro-ene Arylation Reaction of N-Alkoxyenamides for the Synthesis of tert-Alkylamines
11:45 - 12:00 L-3 Rebecca E. Norman, Australia
Synthesis and Reactivity of the Novel Pyrazolo[1,5 b]thiatriazine Ring System
12:00 - 12:15 L-4 Cedric W McCleland, South Africa
DCC/DMAP-Promoted Esterification Reactions in Ionic Liquids and under Solvent-Free Conditions
12:15 - 12:30 L-5
Steen Ingemann Jorgensen, Netherlands
Novel Cinchona alkaloid derivatives as organocatalysts for asymmetric synthesis

Session II
Chair: József Rábai
11:15 - 11:30 L-6 David St C Black, Australia
Synthesis of Indorphyrins and Related Heterocyclic Platforms
11:30 - 11:45 L-7 Ishmael Masesane, Botswana
2’-Hydroxychalcones as Intermediates in the Synthesis of Chromenes
11:45 - 12:00 L-8 Masafumi Ueda, Japan
Regioselective Cyclization of 2-Alkynyl-N-methoxybenzamides
12:00 - 12:15 L-9 Ola K. Al-Sakka, Egypt
2-Substituted Thiophenes: Synthesis, Crystal-Structure and In-Vitro Anti-Tumor Evaluation
12:30 - 14:00 Lunch
Chair: Margaret Brimble
14:00 - 15:00 PL-4 Mark A Rizzacasa, Australia
Total Synthesis: Applications in Structure, Biosynthesis and Biology
15:00 - 15:30 IL-3 Tamás Kálai, Hungary
Synthesis and Applications of Carbo- and Heterocycles  Condensed with Nitroxide Free Radicals
15:30 - 16:00 IL-4
Saverio Florio, Italy
Syntheses Based on Small Ring Heterocycles
16:00 - 16:30 Coffee Break

Short Oral Presentations

Session I
Chair: Tohru Fukuyama
16:30 - 16:45 L-10 Adrien Quintard, France
Dual Iron/Organo-Catalysis for Sustainable Enantioselective Synthesis
16:45 - 17:00 L-11 Ekaterina Budynina, Russia
Ring-Forming Reactions of Donor-Acceptor Cyclopropanes: Cycloaddition vs Annulation
17:00 - 17:15 L-12 Enrico Marcantoni, Italy
Lewis Acid Catalyzed Synthesis for the Preparation of Biologically Active Small Molecules
17:15 - 17:30 L-13 Francisco Alonso, Spain
Multicomponent Synthesis of Heterocycles Catalysed by Supported Copper Nanoparticles
17:30 - 17:45 L-14
Viktor Milata, Slovakia
Ring Transformations of Fused Selenadiazoles
17:45 - 18:00 L-15 Kristína Plevová, Slovakia
Synthesis and Biological Screening of Novel Nucleosides Derived from Trifluoromethoxy-4-Quinolones

Session II
Chair: Kiosey Takasu
16:30 - 16:45 L-16 Ross P. McGeary, Australia
Investigations into the Benzyl-Claisen rearrangement
16:45 - 17:00 L-17 Dibakar C Deka, India
FeCl3.6H2O Catalyzed Water Mediated Facile Domino Synthesis of 5-Alkylidene-/Arylidenebarbituric Acids
17:00 - 17:15 L-18 Hormi Mecadon, India
FeCl3.6H2O Catalyzed Aqueous Media Domino Synthesis of 5-Monoalkylbarbiturates: Water as Both Reactant and Solvent
17:15 - 17:30 L-19 Subarna Jyoti Kalita, India
A Water-Acetic Acid Mediated Raection: Expedient Synthesis of New Benzo[4,5]Imidazo[1,2-A]Pyrimido[4,5-D]Pyrimidine-2,4(1h,3h)-Diones
17:30 - 17:45 L-20 Melinda Fekete, Hungary
A general process for the green and sustainable production of N-alkylimidazoles in flow
17:45 - 18:00 L-21 Rodney A. Fernandes, India
First Stereoselective Total Synthesis of (-)-Asteriscunolide C, a Potent Anticancer Medium Ring Sized Macrolide
 

Tuesday, 01 July 2014

07:30 - 08:45 Registration
Chair: Lutz F. Tietze
08:45 - 09:45
PL-5
Marco A. Ciufolini, Canada
Synthetic Studies on Heterocyclic Natural Products
09:45 - 10:15 IL-5 Anna Trzeciak, Poland

Palladium catalysts in C-C bond forming reactions - mechanistic studies
10:15 - 10:45 IL-6 Kiyosei Takasu, Japan
Discovery of new reactions and utilities of 4-membered carbocyles
10:45 - 11:15 Coffee Break

Short Oral Presentations
Session I
Chair: Tamás Kálai
11:15 - 11:30 L-22 Yoichiro Kuninobu, Japan
Regioselective Trifluoromethylation of N-Heteroaromatic Compounds using BF2CF3 Activator
11:30 - 11:45 L-23 Thomas W Bevan, New Zealand
Colourful azulene-based protecting groups for the protection of carboxylic acids
11:45 - 12:00 L-24 Malek Nechab, France
Transfer of Chirality in Cycloisomerization of Enediynes
12:00 - 12:15 L-25 József Rábai, Hungary
Unusual optical resolution processes for racemic carboxylic acids
12:15 - 12:30 L-26
Ajoy K Banerjee, Venezuela
First Synthesis of 1, 4-Dimethoxy-2-Naphthoxy Acetic Acid

Session II
Chair: Svetlana  Tsogoeva
11:15 - 11:30 L-27 Szabolcs Kovács, Hungary
Application of Aryl Imidazolylsulfonates in Organic Transforamtions
11:30 - 11:45 L-28 Florence Mongin, France
Synergic Mixed Metal 2,2,6,6-Tetramethylpiperido Bases: Wonderful Tools for the Functionalization of Aromatic Heterocycles
11:45 - 12:00 L-29 Robert Tuba, Qatar
Synthesis of Cyclo- and Functionalized Polypentenamers
12:00 - 12:15 L-30 Peter Dalko, France
Light Gated Fast Release Systems
12:15 - 12:30 L-31
Muhammad Azhar Abbas, Pakistan
Synthesis, Characterization and Biological studies of Schiff Base Complexes Derived from Piperazine
12:30 - 14:00 Lunch
14:00 - 16:00 Poster Session
16:00 - 16:30 Coffee Break
Chair: Victor A. Snieckus
16:30 - 17:45 PL-10 Martin D. Burke, United States
the winner of the 2014 Thieme-IUPAC Prize
Making Molecular Prosthetics with a Small Molecule Synthesizer

Wednesday, 02 July 2014

07:30 - 08:45 Registration
Chair: Marco A. Ciufolini
08:45 - 09:45 PL-6 Minoru Isobe, Taiwan
Stereochemical controlled in total synthesis toward Natural Products - Solanoeclepin A nnd Prostaglandin-
09:45 - 10:15 IL-7
Kevin Booker-Milburn, United Kingdom
Photochemical Methods for Complexity Generation
10:15 - 10:45 IL-8 
Krishna P Kaliappan, India
Agonies and Ecstasies in Total Synthesis
10:45 - 11:15 Coffee Break

Short Oral Presentations

Session I
Chair: Hiriyakkanavar Ila
11:15 - 11:30
L-32 Arie Lev Gruzman, Israel
Rational design and synthesis of new peptidomimetic drug candidates for treatment of prostate cancer
11:30 - 11:45 L-33 
Martin Zahel, Germany
Syntheses of Oxygen-Bridged Guaiane Sesquiterpenes Englerin A and Oxyphyllol
11:45 - 12:00 L-34
Alberto Brandi, Italy
Access to Benzo-Fused Lentiginosines
12:00 - 12:15 L-35 
Nicholas J Rudgley, Australia
Total Synthesis of Paecilopyrone A and Phomapyrone B
12:15 - 12:30 L-36
Steve Ludwig, Germany
Synthesis and biocatalytical conversion of new artificial isoprenoids

Session II
Chair:  Saverio Florio
11:15 - 11:30
L-37 Csaba Tömböly, Hungary
Preparation of Semisynthetic Cholesteryl Lipoproteins and their Application in Live Cell Imaging
11:30 - 11:45 L-38
Masahiko Seki, Japan
A New Catalytic System for Ru-Catalyzed C-H Arylation
11:45 - 12:00 L-39 Shigeru Arai, Japan
Pinpoint Cyanation of SP And SP2 Carbons under Nickel Catalysis
12:00 - 12:15 L-40 Takeshi Takeda, Japan
Copper(I)-Promoted Cross-Coupling of Alkenyl and Arylsilanes
12:15 - 12:30 L-41
Damien Bonne, France
Novel Reactivity of 1,2-Dicarbonyls in Organocatalyzed Transformations
12:30 - 14:00 Lunch
14:00 - 16:00 Poster Session
16:00 - 16:30 Coffee Break

Short Oral Presentations
Session I
Chair: Cristina L. L. Chai
16:30 - 16:45 L-42 Takaaki Harada, Japan
Synthetic Studies on Gelsemium Alkaloids
16:45 - 17:00 L-43 Liam J Bromhead, Australia
Enantioselective Synthesis of All Four Stereoisomers of the Strigolactone Mimic GR24
17:00 - 17:15 L-44 
Emily M Boyd, New Zealand
Total Synthesis of Aspergilazine A
17:15 - 17:30 L-45 Marco Buccini, Australia
A 4-Step Synthesis of Radermachol
17:30 - 17:45 L-46 Jingjing Wang, New Zealand
Bestmann Ylide Cascade in the Synthesis of Marine Natural Product (-)-Zampanolide and its Analogues
17:45 - 18:00 L-47 Santosh J. Gharpure, India
Stereoselective Synthesis and Applications of Donor-Acceptor Substituted Cyclopropanes (DACS)
Session II
Chair: Girolamo Cirrincione
16:30 - 16:45 L-48 Hidehiro Sakurai, Japan
Anomalous Efficacy of Bimetallic Au/Pd Nanoclusters  in C-Cl Bond Activation
16:45 - 17:00 L-49 Hiroaki Sasai, Japan
Catalytic Enantioselective Pd(II)/Pd(IV) Reactions Using SPRIX Ligand
17:00 - 17:15 L-50
Fruzsina Szabó, Hungary
Mild, practical methods for the synthesis of aminobenzophenon derivatives via removable group-directed palladium catalyzed C-H activation
17:15 - 17:30 L-51 Tanja Gaich, Germany
Synthetic Expeditions in Indole alkaloid Syntheses
17:30 - 17:45 L-52 
Aaron L Brown, Australia
Total synthesis of ustiloxin D

20:00 - 21:00

Organ Concert

Thursday, 03 July 2014

07:30 - 08:45 Registration
Chair: Jay Siegel
08:45 - 09:45 PL-7 
Max Malacria, France
A journey in radical mediated and transition metal catalyzed polycyclization reaction cascades
09:45 - 10:15 IL-9
Claudio Palomo, Spain
Control of Stereoselectivity in Asymmetric Organic Reactions
10:15 - 10:45 IL-10 Svetlana Tsogoeva, Germany
Asymmetric Synthesis of Nitrogen-Containing Versatile Compounds Through Bifunctional Organocatalysis
10:45 - 11:15 Coffee Break

Short Oral Presentations
Session I
Chair: Stephen B. H. Kent
11:15 - 11:30
L-53 Akihiro Ogura, Japan
One-Pot Glycan Conjugation to Protein via Azaelectrocyclization: Dynamics Analysis of Neoglycoproteins in Live Animal
11:30 - 11:45 L-54 
Gábor Tasnádi, Austria
Nicotinamide-Independent Asymmetric C=C-Bond Reduction by Ene-Reductases
11:45 - 12:00 L-55 Suguru Yoshida, Japan
Molecular conjugation based on enhanced clickability of doubly sterically-hindered aryl azides
12:00 - 12:15 L-56 Ágnes Peragovics, Hungary
Design of Synthetically Accessible Virtual Libraries with Plexus

Session II
Chair: Antal Csámpai
11:15 - 11:30 L-57 Nawal Serradji, France
Design and Synthesis of 3-Isoxazolidone Derivatives as New Chlamydia Trachomatis Growth Inhibitors
11:30 - 11:45 L-58 Fanny J Lombard, Australia
The synthesis of spiroacetals via C-H insertion
11:45 - 12:00 L-59
M. I  Ahmed, Australia
Incrementally Increasing the Flexibility of a Peptide Backbone: Effect on Macrocyclisation Efficiency
12:00 - 12:15 L-60 Marcin Mielczarek, Australia
Synthesis and Biological Activity of Novel Bis-indole Inhibitors of Bacterial Transcription Initiation Complex Formation
12:15 - 12:30 L-61
Pascale Moreau, France
Synthesis of 1,6-dihydropyrazolo[4,3-c]carbazoles and 3,6-dihydropyrazolo[3,4-c]carbazoles with Pim kinase inhibitory potencies
12:30 - 14:00 Lunch

Chair: Minoru Isobe
14:00 - 14:30 IL-11
Christina LL Chai, Singapore
Synthetic approaches to nature-inspired compounds for drug discovery
14:30 - 15:00 IL-12 
Ila Hiriyakkanavar, India
Molecular Diversity Generation Through Novel Organosulfur Synthons: Versatile Templates for Heterocycle Synthesis
15:00 - 15:30 Coffee Break

Short Oral Presentations
Session I
Chair: Tamás Patonai
15:30 - 15:45 L-62 Rakesh Kumar, India
Non-Biomimetic Oxidation of 1,4-Dihydropyridines: New Methodology for the Synthesis of Bicyclic Heterocycles
15:45 - 16:00 L-63 Dattatraya H Dethe, India
Biomimetic Total Syntheses of the Borreverine, Caulindole and Flinderole Alkaloids
16:15 - 16:30 L-64 Imre Hegedüs, Hungary
Grafting from" synthesis of organic capsule around single protein molecules
16:30 - 16:45 L-65
Vasoulla N Moussa, Australia
Isolation and Chemistry of Compounds Found in the Western Australian Plant Dodonaea Ceratocarpa
16:45 - 17:00 L-66
Amélia P. Rauter, Portugal
An Efficient Synthetic Route to Antimicrobial Deoxy Glycosides

Session II
Chair: Krishna P. Kaliappan
15:30 - 15:45 L-67
Fabrice Anizon, France
Dipyrrolo[3,4-a:3,4-c]carbazoles as kinase inhibitors
15:45 - 16:00 L-68 Krisztina Kónya, Hungary
Synthesis of Flavonoid – and Chromonoid-D-Glucopyranoside Hybrids with Unsaturated Carbon Bridge by Palladium Catalysed Cross-coupling Reactions
16:15 - 16:30 L-69 Antal Csámpai, Hungary
Synthesis of novel planar chiral ferroceno-fused heterocycles of biological relevance
16:30 - 16:45 L-70
Mohammad M Ghanbari, Iran
An Efficient One-Pot Synthesis Of Novel Imidazoles
16:45 - 17:00 L-71
Qingchao Liu, China
Synthesis and biological evaluation of N-linked sugar-substituted oleanolic acid derivatives as PTP1B inhibitors

20:00 - 22:00


Conference Dinner


Friday, 04 July 2014

07:30 - 08:45 Registration
Chair: Max Malacria
08:45 - 09:45 PL-8 
Johann H Mulzer, Austria
Last reflections on total synthesis
09:45 - 10:15 IL-13
Girolamo Cirrincione, Italy
Isoindolo[2,1-a]Quinoxalin-6-Imines: In Vitro and In Vivo Antitumor Activity and G-Quadruplex Stabilizing Effect
10:15 - 10:45 Coffee Break

Chair: Johann Mulzer
10:45 - 11:45 PL-9 Eusebio Juaristi, Mexico
Recent advances in asymmetric synthesis under solvent-free reaction conditions

11:45 - 12:15

Closing with Poster Prize Award

12:15 - 14:00

Lunch

 


POSTER PRESENTATIONS



P-01 Mehlika Dilek Altintop, Turkey
Synthesis and In Vivo Evaluation of 1,3,5-Trisubstituted Pyrazolines as Antidepressant-Like Agents
P-02 Norihito Arichi, Japan
Synthesis of Steroid Derivatives Bearing a Small Ring  for the Conformational Fixation of D-Ring Side Chain
P-03 Gülgün Ayhan-Kilcigil, Turkey
Synthesis and Evaluation of Antioxidant Activities of Novel 1,3,4-Oxadiazole and Imine Containing 1H-Benzimidazoles
P-04 Aigerim Kenzhebekovna Badanova, Kazakhstan
Synthesis of Polymer Film on Cellulosic Fiber for Imparting Hydrophobic Properties
P-05 Norah Bennamane, Algeria
Reactivity of Enaminones:  Synthesis of Amino  1, 5- Benzodiazepines, Benzotriazoles and N, N'-Bis(2- Aminophenyl)But-2-Enediamide System
P-06 Eileen Bette, Germany
First asymmetric total synthesis of the natural fungicide Hygrophorone B12
P-07 Dattatry Bhosale, Czech Republic
Henry Recation Catalysed by Recoverable Enantioselective Catalysts Based on Copper(Ii) Complexes of a-Methoxypoly(Ethylene Glycol)-B-Poly(L-Glutamic A
P-08 Gomotsang Bojase, Botswana
Exploratory Chemistry Of Dendralenes
P-09
Jana Boržiková, Slovakia
Reactivity, Synthesis and Structure Reactivity of  New 3-Benzoylthiophen derivatives as Potential Biologically Active Compounds and Novel Opto-electronic Materials
P-10 Kamal H. Bouhadir, Lebanon
Preparation and Biological Evaluation of Acylydrazono-Carbanucleosides for Diabetic Nephropathy
P-11 Diego Carnaroglio, Italy
Nanomaterial surface functionalization and grafting under microwave irradiation
P-12 Raju Cheerlavancha, Australia
Synthesis of Alpha,Beta,Gamma-Trifluoro-Delta-Amino Acids
P-13 Jeonghun Cho, South Korea
Dynamic Kinetic Resolution of Boron-Containing Secondary Alcohols
P-14 Daniel Frazer Chorley, New Zealand
Synthetic studies towards pinnatifinoside C & D
P-15 Jacek Chrzanowski, Poland
Thioureas Derived From Optically Active a-(2-Pyridyl)ethylamine
P-16 HsiangYu Chuang, Taiwan
Synthetic Studies toward Solanoeclepin A
P-17 Wojciech Ciesielski, Poland
Functionalization Carbon Nanotubes by Compounds with a Sulphur and Phosphorous Stereogenic Heteroatoms
P-18 Robert Alexander Clegg, Australia
Development of inhibitors for N-Myristoyltransferase
P-19 Paulo Coelho, Portugal
Preparation of Organic/Inorganic Hybrid Matrices Doped with Photochromic Naphthopyrans
P-20 Philip G. E. Craven, United Kingdom
Natural Product-Inspired Libraries for the Exploitation in the European Lead Factory
P-21 Ruth Deme, Hungary
D-Annelated Steroids through Type 2 Tert-Amino Effect
P-22 Nahide Gulsah Deniz, Turkey
An Efficient One-Pot Multicomponent Synthesis of Naphthoquinone Compounds
P-23 Nahide Gulsah Deniz, Turkey
The Vinylic Substitution Reactions of Polyhalogenated Nitrodiene with Thiol and Amine Derivatives
P-24 Krzysztof Dudzinski, Poland
Acetone Cyanohydrin as a Safe Cyanide Source in the Enantioselective Organocatalytic Strecker Reaction
P-25 Gábor Durkó, Hungary
On the mechanism of the solvent-induced cubane - cuneane rearrangement
P-26 Mohamed A El-borai, Egypt
Eco-Friendly Preparation of 4-Bromo Pyrazolone and the Study of its Reactivity by Microwave and Classical Techniques
P-27 Gergely Farkas, Hungary
Novel aminoalkyl-phosphine ligands and their application in the asymmetric synthesis of chiral synthons
P-28 Gabriella Fiser, Hungary
Semisynthesis of Fluorescent Lipoprotein Derivatives for Studying Membrane-associated Proteins
P-29 Emese Gal, Romania
Synthesis of novel phenothizinyl/phenyl mono and di-nitrones, EPR and DNA interaction study
P-30 Ali Gharib, Iran
Catalytic Synthesis of Pyrano- And Furoquinolines using Nano Silica Chromic Acid (Nano Sca) at Room Temperature
P-31 Ali Gharib, Iran
A Novel and Facile One-Pot Synthesis Of Pyrazolo[3,4-D]Pyrimidine-6-Thiol and Pyrazolo[3,4-D]Pyrimidin-6-Ol Derivatives using Nanoparticles of Nax Zeo
P-32 Michael Ghobrial, Austria
Exploration of C-H and N-H Bond Functionalization Towards 1-(1,2-Diarylindol-3-Yl)-Tetrahydroisoquinolines
P-33 Zsombor Gonda, Hungary
In Situ Generated Trifloromethyl Alkylborate Salts - a Simply Method for Copper Catalyzed Trifluoromethylation of Aromatic and Heteroaromatic Iodide
P-34 Gergely Gulyás, Hungary
Carotenoid-flavonoid hybrids
P-35 Hyun-Joon Ha, South Korea
Synthesis Of Hyacinthacinie A1 from Chiral Aziridine
P-36 Ales Halama, Czech Republic
Convenient Synthesis of Rivaroxaban from (S) Epichlorhydrin
P-37 Lamouri Hammal, Algeria
Synthesis and biological evaluation of some benzodiazepine structures
P-38 Jiayun He, Hong Kong
Investigation on Intramolecular (4+3) Cycloadditions of Pyrrole and the Synthetic Application Towards Type II Galbulimima Alkaloids
P-39 Martin Hennum, Norway
Nitrogen substituted quaternary stereocenters from the Overman rearrangement and the allyl cyanate-to-isocyanate rearrangement
P-40 Day-Shin Hsu, Taiwan
Total Synthesis of (+/-)-Nidemone
P-41 Judit Huber, Hungary
Syntheses of 16-acylamino derivatives in the 13?-estrone-series and their antiproliferative activities
P-42 Steen Ingemann Jorgensen, Netherlands
Synthesis of Quinuclidines by Silver Catalysed Hydroamination
P-43 Yuta Ito, Japan
Direct Synthesis of Benzofuro[2,3-b]pyrroles by a Domino Reaction Involving a Radical Addition and [3,3]-Sigmatropic Rearrangement
P-44 Darvin S. Ivanov, Bulgaria
Synthesis, geometry optimization and cytotoxic activity of new bromo-salicylaldehyde hydrazones
P-45 Eun-Sil Kang, South Korea
Studies toward efficient conversion of biomass into furanic platform chemicals
P-46 Dae Young Kim, South Korea
Enantioselective Organocatalytic Oxidative Enamine Catalysis/1,5-Hydride Transfer/Cyclization Sequences: Asymmetric Synthesis of Tetrahydroquinolines
P-47 Krisztina Knapp, Hungary
Thiol-Specific Fluorescent Labels for Monitoring UV Mediated Disulfide Scission
P-48 László Kocsis, Hungary
Synthesis Of Novel Ferrocene Containing Cinchona Alkaloid Derivatives
P-49 Moo-hyun Koh, South Korea
Functional Group Transformations of Vegetable Oils and their Applications to Polyamide Monomers
P-50 Zoltán Kondor, Hungary
Synthesis of New Furanoside-Chromonoid and -Flavonoid Hybrids with Heck Reaction
P-51 Dóra Kovács, Hungary
Efficient approach to novel ring-condensed steroidal isoxazolines by 1,3-dipolar cycloaddition
P-52 Dorota Krasowska, Poland
Cyclic Chiral Phosphonic Acid Derivatives Based on Phenol Residue-Containing Chiral Auxiliaries: Syntheses and Reactivity
P-53 Damian Kulawik, Poland
The Search for New Chiral Ionic Liquids with  Tetracoordinated and/or Hypervalent Heteroatoms
P-54 Yusuke Kuroda, Japan
Synthesis of 2,3,4,5-tetra-substituted pyrroles via a base-promoted double Michael reaction of oxime-enoates
P-55 Hee-Yoon Lee, South Korea
Total synthesis of crinipellin A
P-56 Hee-Yoon Lee, South Korea
Total Synthesis of Waihoensene
P-57 Jusuk Lee, South Korea
Dynamic Kinetic Resolution of Diaryl Carbinols
P-58 László Csaba Lengyel, Hungary
Synthesis of Condensed Heterocycles by the Gould-Jacobs and Conrad-Limpach Reaction in a Novel Three-Mode Pyrolysis Reactor
P-59 Jesse Ling, Hong Kong
Diastereoselective Friedel-Crafts alkylation of epoxy enolsilanes
P-60 Klára Lövei, Hungary
Continuous Flow Synthesis of Novel Heterocycles with Druglike Properties
P-61 Ramaiyan Manikannan, Czech Republic
Synthesis and Properties of Push–Pull–Push Chromophores  Based on 3,4-Dinitrothiophene
P-62 Erzsébet Mernyák, Hungary
Preparation of Novel Cytostatic D-Secoestrone Conjugates
P-63 Ádám Mészáros, Hungary
Synthesis of new benzoxazine derivatives via copper catalyzed oxidative cyclization utilizing arylethynyl pivalanilides and diaryliodonium salts
P-64 Adam G Meyer, Australia
An iterative modelling and modular synthetic approach to tercyclic alpha-helix mimetics with measured aqueous solubility
P-65 Kristina Mickevičiene, Lithuania
Synthesis And Properties of 3-(6,11-Dioxo-6,11-Dihydro-12h-Benzo[B]Phenoxazin-12-Yl)Butanoic Acid Derivatives
P-66 Kristina Mickevičiene, Lithuania
New S,N-Containing Heterocycles Based on Benzoylthioureas of 9,10-Anthraquinones
P-67 Marcin Mielczarek, Australia
Synthesis of New Heterocyclic Structures Based on Indoles, Oxadiazoles and Thiadiazoles
P-68 Toshifumi Miyazawa, Japan
Boronic Mannich Reaction Using N-Pyruvoylamino Acid Derivatives as Oxo Components
P-69 Pravinkumar H Mohite, Czech Republic
Optically Active Amines Bearing Benzo[D]Imidazole and a-Amino Acid Pendants and their Application in Asymmetric Aldol Reaction
P-70 Florence Mongin, France
Access to Functionalized Azoles and Polyazoles through Deprotometalation-Iodination followed by Transition Metal Catalyzed Reactions
P-71 Pascale Moreau, France
Synthesis of 1,6-dihydropyrazolo[4,3-c]carbazoles and 3,6-dihydropyrazolo[3,4-c] carbazoles with Pim kinase inhibitory potencies
P-72 Gergő Mótyán, Hungary
Stereoselective Synthesis of New Androstene-Fused Arylpyrazolines as Potent Antiproliferative Agents
P-73 Vasoulla N Moussa, Australia
Isolation and Chemistry of Compounds Found in Dodonaea Ceratocarpa
P-74 Štefan Možina, Slovenia
Activation of nitration of aromatic compounds by template catalysis
P-75
Ion Neda, Romania
Bifunctional Derivatives of the Isophosphoramide Mustard
P-76 Bellara Nedjar-Kolli, Algeria
An Efficient Synthesis of Electroactive 1,5-Benzodiazepines
P-77 Bellara Nedjar-Kolli, Algeria
Synthesis of Thiosemicarbazones and their Cyclisation to 4-Thiazolidinones
P-78 Anikó Nemes, Hungary
Synthesis and Application of Chiral (Nonafluoro-Tert-Butoxy)Carboxylic Acids
P-79 Péter Nemes, Hungary
New synthetic route to fused pyrimidines
P-80 Akiko Okamoto, Japan
Crystal Structure Study of Non-Coplanarly Organized Accumulating Aromatic Rings Molecules: Spatial Organization of C,C,N-Triaryl Substituted Imines
P-81 Ahmet Özdemir, Turkey
Chloro-Substituted Pyrazolines As Antidepressant Agents
P-82 Dávid Pajtás, Hungary
Selective Suzuki and Buchwald-Hartwig reaction of 6,7- and 6,8-dibromoflavones
P-83 Máté Papp, Hungary
Aminocarbonylation of iodobenzene in the presence of SILP-palladium catalysts
P-84 Britt Paulsen, Norway
Synthesis of bioactive ent-ageloxime D, and a terpenoid analog
P-85 Dijana Pešić, Croatia
Novel Macrolide Inspired Macrocyclic Library
P-86 Bálint Pethő, Hungary
Palladium-Catalyzed Methoxylation of Aromatic Chlorides with Borate Salts
P-87 Karolina Piecyk, Poland
Synthesis of 1,2,3-Triazole Containing Dinucleotide TMG Cap Analogues for Binding Studies with Snurportin-1
P-88 Falko Pippig, Czech Republic
Imidazolium Based Donor-Acceptor Chromophores
P-89 Mária Polyák, Hungary
Study of Can Mediated Transformations 1-C-Substituted Glycals
P-90 Mihaly Posa, Serbia
Wittig Reaction (with Ethylidene Triphenylphosphorane) of Oxo-Hydroxy Derivatives of 5ß-Cholanic Acid: Novel Cholesterol Solubilisators
P-91 Oleg A. Rakitin, Russia
One-Pot Conversion of Fused 1,2,5-Thiadiazoles into 1,2,5-Selenadiazoles
P-92 Isaiah D I Ramaite, South Africa
Suzuki Reaction in the Synthesis of 6-Arychromone-3-carbaldehydes and derivatives
P-93 Karl Rautschek, Germany
Studies Towards The Synthesis Of Scabrosin A
P-94 Attila Remete, Hungary
Fluorinations of Highly Functionalized Alicyclic Beta-Amino Acids
P-95 Young Rhee, South Korea
Metal-catalyzed asymmetric hydroamination of alkoxyallene: Development and Application
P-96 Fumie Sakurai, Japan
Development of an Aquacatalytic System Based on the Vesicle Formation of an Amphiphilic NNC-Pincer Palladium Complex
P-97 Shohei Sato, Japan
One-pot Phenylation/Addition Reaction to N-Alkoxyenamines
P-98 M. Cigdem Sayil, Turkey
Electro- and Photochemical Properties of Naphthoquinone Derivatives
P-99 M. Cigdem Sayil, Turkey
Synthesis and Molecular Structures of Heteroatom Substituted Quinone Compounds
P-100 Katharina M. Schragl, Austria
Synthesis of doping-relevant arylpropionamide-derived SARM metabolites
P-101 Mónika Sebestyén, Hungary
NaBH4 – A Novel Modest Method For The Deprotection Of Nw-Nitro-Arginine
P-102 Maiju Soikkeli, Finland
Synthesis of 2,2,6,6-teraethylpiperidin-1-oxyl-4-yl-ß-D-glucopyranoside, a water soluble stable nitroxide radical
P-103 P.B. Solanke, Czech Republic
Synthesis  and UV/VIS Study of T-Shaped Push-Pull Chromophores
P-104 Sebastian Steiner, Austria
Towards Biomimetic Total Synthesis of Elisabethin A
P-105 Magne Sydnes, Norway
Enantioselective Total Synthesis of Trans-1,2-Diol Metabolites of 3 and 4.Ring PAHs
P-106 Johanna Szabó, Hungary
Synthesis of novel antiproliferative D-secoalkynes of 13a- and 13b-estrone and their heterocyclic derivatives
P-107 Nikoletta Szabó, Hungary
Synthesis of Some 17-Picolyl and 17-Picolinylidene Androstane Derivatives and their Inhibitory Effect against the D5-3ß-HSD ...
P-108 Eszter Szennyes, Hungary
Synthesis of 1-C-Hetaryl-Glucals for The Inhibition of Glycogen Phosphorylase
P-109 Gábor Szilvágyi, Hungary
Twisted dirhodium complexes of natural and modified amino acids: synthesis and structure determination using chiroptical methods (ECD, VCD)
P-110 Aliz Szloszár, Hungary
Organocatalysis in flow: solid supported peptide catalyzed asymmetric α-amination of aldehydes
P-111 Péter Szuroczki, Hungary
Synthesis and Study of New Parp Inhibitors Modified with Niroxides or Nitroxide Precursors
P-112
Nripendra N Talukdar, India
An Efficient Biomass-derived Heterogeneous Base Catalyst for Transesterification of Vegetable Oils to Biodiesel
P-113 Julia Timmel, Germany
Application of a Temporary Thiophenyl Group for the Enantioselective Synthesis of Codeine
P-114 Chisato Tsuruoka, Japan
Synthesis of HOMSi Reagents by Palladium-catalyzed Silylation of Bromoarenes using Disilanes
P-115 József Tukacs, Hungary
Platform chemicals from biomass, improved catalyst system for the reduction of levulininc acid to gamma-valerolactone
P-116 Meral Tuncbilek, Turkey
Novel 6-(4-Substituted Piperazine-1-Yl)-9-(ß-D-Ribofuranosyl)Purine Derivatives: Synthesis and Cytotoxic Activity on Selected Human Cancer Cell Lines
P-117 Ahmet Tutar, Turkey
Synthesis of Bromo Substituted 11H-indeno[1,2-b]quinolin-10-ylamine Derivatives via Friedländer Reaction
P-118 Marietta Vágvölgyiné Dr. Tóth, Hungary
Xylose Derived Inhibitors of Glycogen Phosphorylase
P-119 Marietta Vágvölgyiné Dr. Tóth, Hungary
A New Route for The Synthesis of Asymmetric 3,5-Disubstituted-1,2,4-Triazoles and 3-C-Glycosyl-5-Aryl-1,2,4-Triazoles
P-120 Gábor Varró, Hungary
An expedient stereoselective total synthesis of (±)-trans-dihydro-narciclasine
P-121 Daniel Végh, Slovakia
Strategies, Design And Synthesis of Highly Electroluminescent Devices made with a Conveniently Synthesised 2-Thienyl- 2´-(1h-Pentafluorophenyl)P
P-122 Veronica Tecchio, Australia
Synthesis of Variolin B Analogs: Novel Inhibitors of Alternative Splicing Kinases
P-123 Elena V. Villemson, Russia
Ring Opening of Donor-Acceptor Cyclopropanes with Azide Ion as an Essential Step in N-Heterocycles Construction
P-124 Jakob K K Wahlander, Norway
Synthesis Directed Towards Asmarine Fragments and Development of Lewis Acid Diels-Alder Catalysts
P-125 Agata M Wrześniewska, Poland
Synthesis and Antibacterial Activity of Schiff Bases and Amines Derived from Alkyl 2-(2-Formylphenoxy)alkanoates
P-126 Sayaka Yoshiwaka, Japan
Spatial Organization of Peri-Aroylnaphthalene Derivatives: Discrimination of X-Ray Crystal Structure-Determinig Interactions
P-127 Árpád Balázs, Hungary
Silver(I)-catalyzed synthesis of 2- and 3-substituted quinolines and naphthiridines
P-128 Ramóna Madácsi, Hungary
Investigation of SNAr reactions of 2-(2,6-diisopropylphenyl)-4,5,6,7-tetrafluoroisoindoline-1,3-dione with amines